Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_02123
Ion Channel
Neuronal acetylcholine receptor subunit alpha-9/alpha-10
Peptide Function
Antagonist
Gene Name
CHRNA9/CHRNA10
Activity Data (nM)
IC50
5.2 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
GCCSDPRCRYRCR
Peptide UniProt Accession
UniParc
UPI0000D8554A
Peptide Synonyms/Alias
alpha-RgIA
Peptide Species
Conus regius (Crown cone)
Peptide Name
Alpha-conotoxin RgIA
CAS Number
876728-23-3
Experimental Conditions
pH
pH 7.1 to 7.5
Holding Potential (mV)
−70 mV
Temperature
22 °C
Test Method
Patch-clamping
Test Species
Not specified
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
nAChRs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available